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Cat. No. Product Name Target Signaling Pathways
TP2073L BigLEN (mouse) acetate

BigLEN (mouse) acetate (501036-69-7 Free base)

GPR Endocrinology/Hormones; GPCR/G Protein
BigLEN (mouse) acetate 是一种有效的、选择性的孤儿 G 蛋白偶联受体 171 (GPR171) 激动剂,Kd 为 ~0.5 nM。
TP2073 BigLEN(mouse)

BigLEN (mouse)

GPR171 agonist. ProSAAS-derived neuropeptide. Regulates food intake in mice. Inhibits the release of glutamate onto parvocellular neurons of the paraventricular nucleus in a process dependent upon activation of postsynaptic G proteins.
TP2074 BigLEN(rat)

BigLEN (rat)

Potent GPR171 agonist (EC50 = 1.6 nM). ProSAAS-derived peptide. Regulates body weight in mice and promotes the outgrowth of neurites in Neuro2A cells.
T76046 BigLEN(rat) TFA

BigLEN(rat)是一种有效的GPR171激动剂,其EC50为1.6 nM。
T82885 BigLEN(mouse) TFA

BigLEN(mouse) TFA 是一种GPR171激动剂,同时也是源自proSAAS的神经肽。该化合物调节小鼠的食物摄入,并且依赖于突触后G蛋白的激活,抑制谷氨酸释放到下丘脑室旁核的旁核细胞上。

化合物

BigLEN (mouse) acetate
Cat.No: TP2073L
Synonym: BigLEN (mouse) acetate (501036-69-7 Free base)
Target: GPR
BigLEN(mouse)
Cat.No: TP2073
Synonym: BigLEN (mouse)
Target:
BigLEN(rat)
Cat.No: TP2074
Synonym: BigLEN (rat)
Target:
BigLEN(rat) TFA
Cat.No: T76046
Synonym:
Target:
BigLEN(mouse) TFA
Cat.No: T82885
Synonym:
Target:
TargetMol Loading
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