Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2071L |
Bay 55-9837 acetate
|
Glucagon Receptor | GPCR/G Protein |
Bay 55-9837 acetate 是一种有效且高度选择性的 VPAC2 激动剂 (Kd = 0.65 nM),可用于 2 型糖尿病研究。 | |||
TP2071 |
Bay 55-9837
|
||
Selective VPAC2 receptor agonist (EC50 values are 0.4, 100 and >1000 nM for VPAC2, VPAC1 and PAC1, respectively in a cAMP accumulation assay; IC50 values are 60, 8700 and >10000 nM for VPAC2, VPAC1 and PAC1, respectively in a competition binding assay). S |