Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2375 |
BX471
BX 471,BX-471,ZK-811752 |
CCR | Immunology/Inflammation; Microbiology/Virology |
BX471 (BX 471) 是可口服的非多肽 CCR1选择性拮抗剂,Ki 值为 1 nM,对其选择性是对 CCR2、CCR5 和 CXCR4 的 250 倍。 | |||
T14845 |
BX471 hydrochloride
ZK-811752 hydrochloride |
Others | Others |
BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist (Ki: 1 nM for human CCR1). It shows 250-fold selectivity for CCR1 over CCR2, CCR5, and CXCR4. |