Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T38507 |
Renzapride
BRL 24924 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Renzapride (BRL 24924) 是一种混合 5-羟色胺 4 型 (5-HT4) 激动剂和 5-HT3 受体拮抗剂。Renzapride 可用于研究以便秘为主的肠易激综合征(C-IBS)。 | |||
T72809 |
(S)-Renzapride
(S)-BRL 24924 |
||
(S)-Renzapride ((S)-BRL 24924) 是 Renzapride 的异构体。Renzapride 是一种 5-HT4受体激动剂,Ki 值为 115 nM。Renzapride 还是一种5HT2b 和5HT3受体拮抗剂。Renzapride 可用于便秘型肠易激综合征(C-IBS)的研究。 | |||
T28517 |
Renzapride hydrochloride
BRL-24924,ATL1251,ATL-1251,Renzapride HCl,AZM-112 |
||
Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors. |