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Cat. No. Product Name Target Signaling Pathways
T61318 BRD4 Inhibitor-20

Epigenetic Reader Domain Chromatin/Epigenetic
BRD4 Inhibitor-20是一种有效的溴结构域蛋白4(BRD4)抑制剂,具有口服活性。BRD4 Inhibitor-20在癌细胞系中具有抗增殖活性,并被用于各种癌症的研究,如结肠癌。
T64117 BRD4-BD1-IN-2

Epigenetic Reader Domain Chromatin/Epigenetic
BRD4-BD1-IN-2 是一种具有选择性和有效性的 BRD4-BD1 抑制剂,IC50 值为 2.51 µM ,是对 BRD4-BD2 抑制活性的 20 倍。BRD4-BD1-IN-2 可用于研究心血管疾病和癌症相关疾病。
T38381 CAY17c

CAY17c is an inhibitor of bromodomain-containing protein 4 (BRD4; IC50= 0.71 μM), as well as class I histone deacetylases (HDACs; IC50s = 0.046, 0.058, 0.075, and 0.167 μM for HDAC1, -2, -3, and -8, respectively) and class IIb HDACs (IC50s = 0.073 and 0.923 μM for HDAC6 and HDAC10, respectively).1It is selective for these enzymes over BRD2, -3, and -T (IC50s = >20 μM for all), as well as over HDAC4, -5, -7, -9, and -11 (IC50s = >10 μM for all). CAY17c inhibits the proliferation of HCT116, SW620,...

化合物

BRD4 Inhibitor-20
Cat.No: T61318
Synonym:
Target: Epigenetic Reader Domain
BRD4-BD1-IN-2
Cat.No: T64117
Synonym:
Target: Epigenetic Reader Domain
CAY17c
Cat.No: T38381
Synonym:
Target:
TargetMol Loading
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