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Cat. No. Product Name Target Signaling Pathways
T14678 BMS-819881

P450 Metabolism
BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a Ki of 7 nM and it also is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
T71265 BMS-830216

BMS-830216 is a nonbasic melanin hormone receptor 1 antagonist and a prodrug of BMS-819881.

化合物

BMS-819881
Cat.No: T14678
Synonym:
Target: P450
BMS-830216
Cat.No: T71265
Synonym:
Target:
TargetMol Loading
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