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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T15049 Daltroban

BM-13505,SKF 96148

PPAR DNA Damage/DNA Repair; Metabolism
Daltroban (SKF 96148) (BM-13505) 是选择性和特异性的血栓素 A2 (TXA2) 受体拮抗剂。Daltroban 可以增加血管平滑肌细胞内钙。Daltroban 显示对再灌注损伤的保护作用。
T36539 Nocardamine

Nocardamine is a ferrioxamine siderophore that has been found inStreptomycesand has diverse biological activities.1,2,3,4It chelates iron in a chrome azurol S assay (IC50= 9.9 μM).1Nocardamine inhibitsM. smegmatisandM. bovisbiofilm formation (MIC = 10 μM for both), an effect that can be reversed by iron.2It is cytotoxic to T47D, SK-MEL-5, SK-MEL-28, and RPMI-7951 cancer cells (IC50s = 6, 18, 12, and 14 μM, respectively).3Nocardamine also induces morphological changes in BM-N4 insect cells.4 1.Lo...

化合物

Daltroban
Cat.No: T15049
Synonym: BM-13505,SKF 96148
Target: PPAR
Nocardamine
Cat.No: T36539
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T0480 Doxofylline

Doxophylline,多索茶碱

PDE; Adenosine Receptor GPCR/G Protein; Metabolism; Neuroscience
Doxofylline (Doxophylline) 是腺苷 A1 受体拮抗剂,且能抑制磷酸二酯酶 IV,用于治疗哮喘。

天然产物

Doxofylline
Cat.No: T0480
Synonym: Doxophylline,多索茶碱
Target: PDE, Adenosine Receptor
TargetMol Loading
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