Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1442 |
Pizotifen
Pizotyline,BC-105,苯噻啶 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Pizotifen (Pizotyline) 是5-HT2受体的有效拮抗剂,并对5-HT1C 有高亲和力。它是一种强血清素和色胺拮抗剂,具有较弱的抗胆碱能、抗组胺和抗激肽作用,还具有镇静和刺激食欲的特性。 | |||
T0225 |
Pizotifen Malate
Pizotyline (malate),BC-105 (malate),BC-105,苯噻啶苹果酸盐 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Pizotifen Malate (BC-105 malate) 是5-HT2受体的拮抗剂,对5-HT1C 有高亲和力。 |