Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13467 |
(±)-Enitociclib
(±)-BAY-1251152 |
CDK | Cell Cycle/Checkpoint |
(±)-Enitociclib ((±)-BAY-1251152) 是 BAY-1251152 的外消旋混合物。BAY-1251152 是一种高度选择性的 PTEF/CDK9抑制剂。 | |||
T70387 |
CCCTP
|
||
CCCTP is a potent inhibitor of the 11β-HSD-1 enzyme with reduced pregnane-X receptor (PXR) transactivation activity. | |||
T70388L |
(R)-Enitociclib
|
CDK | Cell Cycle/Checkpoint |
(R)-Enitociclib 是 BAY-1251152的一个对映体,是 CDK9 抑制剂,具有抗癌活性。 |