Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T67927 |
BAY-069
|
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
BAY-069 是一种抑制剂。BAY-069对支链氨基酸转氨酶 1 (BCAT1)具有抑制作用(IC50:31 nM ,对支链氨基酸转氨酶 2 (BCAT2) 具有抑制作用(IC50 :153 nM)。BAY-069 是一种新型(三氟甲基)嘧啶二酮类化学探针, 可用于抗癌研究。 | |||
T69518 | BAY-771 | ||
BAY-771 is a negative control of BAY-069, BAY-069 is a BCAT1/2 Inhibitor and Chemical Probe. BAY-069 displays high cellular activity and very good selectivity. BAY-069 displays high cellular activity. Its overall in vivo pharmacokinetic profile and its selectivity in various in vitro panels suggest that BAY-069 is suitable for in vivo experiments. | |||
T78148 |
BAY-252
|
Others | Others |
BAY-252为一种高效的BCAT1及BCAT2 (支链氨基酸转氨酶 1 和 2) 抑制剂,其IC50均值为2 μM。作为化学探针,BAY-252亦适用于癌症研究领域。 |