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Cat. No. Product Name Target Signaling Pathways
T67927 BAY-069

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
BAY-069 是一种抑制剂。BAY-069对支链氨基酸转氨酶 1 (BCAT1)具有抑制作用(IC50:31 nM ,对支链氨基酸转氨酶 2 (BCAT2) 具有抑制作用(IC50 :153 nM)。BAY-069 是一种新型(三氟甲基)嘧啶二酮类化学探针, 可用于抗癌研究。
T69518 BAY-771

BAY-771 is a negative control of BAY-069, BAY-069 is a BCAT1/2 Inhibitor and Chemical Probe. BAY-069 displays high cellular activity and very good selectivity. BAY-069 displays high cellular activity. Its overall in vivo pharmacokinetic profile and its selectivity in various in vitro panels suggest that BAY-069 is suitable for in vivo experiments.
T78148 BAY-252

Others Others
BAY-252为一种高效的BCAT1及BCAT2 (支链氨基酸转氨酶 1 和 2) 抑制剂,其IC50均值为2 μM。作为化学探针,BAY-252亦适用于癌症研究领域。

化合物

BAY-069
Cat.No: T67927
Synonym:
Target: Reactive Oxygen Species
BAY-771
Cat.No: T69518
Synonym:
Target:
BAY-252
Cat.No: T78148
Synonym:
Target: Others
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