Cat. No. | Product Name | Target | Signaling Pathways |
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T21787 |
B-HT 933 dihydrochloride
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Azepexole (B-HT 933) dihydrochloride 是一种有效的选择性α 2肾上腺素受体激动剂,对 α2A-、α2B- 和 α2C- 肾上腺素受体亚型的 pKi 分别为 8.3、7.6 和 7.5。Azepexole dihydrochloride 引起浓度依赖性的蠕动收缩抑制,IC50值为 78.72 nM。 | |||
T69367 |
Azepexole
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Azepexole is a selective α2-adrenoceptor agonist that exhibits greater than 300-fold selectivity for the α2-adrenoceptor over the α1-adrenoceptor. | |||
T21787L |
Azepexole hydrochloride
4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1) |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) 是一种具有麻醉作用的强效α2-肾上腺素受体激动剂。 |