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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T36539 Nocardamine

Nocardamine is a ferrioxamine siderophore that has been found inStreptomycesand has diverse biological activities.1,2,3,4It chelates iron in a chrome azurol S assay (IC50= 9.9 μM).1Nocardamine inhibitsM. smegmatisandM. bovisbiofilm formation (MIC = 10 μM for both), an effect that can be reversed by iron.2It is cytotoxic to T47D, SK-MEL-5, SK-MEL-28, and RPMI-7951 cancer cells (IC50s = 6, 18, 12, and 14 μM, respectively).3Nocardamine also induces morphological changes in BM-N4 insect cells.4 1.Lo...

化合物

Nocardamine
Cat.No: T36539
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T14329 Ascamycin

Nucleoside Antimetabolite/Analog; Others; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ascamycin 是一种由链霉菌属产生的 5'-O-磺酰胺核糖核苷抗生素,对黄单胞菌类显示出选择性的抗菌活性,对柠檬黄单胞菌、口蹄疫黄单胞菌和噬菌体具有抑制作用,MIC 值分别为0.4μg/mL、12.5μg/mL 和12.5μg/mL。

天然产物

Ascamycin
Cat.No: T14329
Synonym:
Target: Nucleoside Antimetabolite/Analog, Others, Antibacterial, Antibiotic
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