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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T73586 Anticonvulsant agent 2

Others Others
Anticonvulsant agent 2 是一种有效的口服活性抗惊厥剂,在耐药性癫痫模型中显示出抗癫痫活性。
T10027 Anticonvulsant agent 1

4-(2,2-Difluoroethenyl)-α-ethyl-2-oxo-1-pyrrolidineacetamide

Others Others
Anticonvulsant agent 1 is an anticonvulsant compound.
T12156 N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea

Others Others
N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea 是一种抗惊厥剂,对广泛强直和部分性发作挛性具有潜在的研究价值。
T22509 3-Methyl-GABA

Others Others
3-Methyl-GABA 是一种有效的GABA 氨基转移酶激活剂。3-Methyl-GABA 能与 GABAA 受体 (GABAaR) 结合。3-Methyl-GABA 能够激活 L-谷氨酸脱羧酶 (GAD),表现出抗惊厥作用。
T60492 Lamotrigine hydrate

Lamotrigine hydrate 是口服有效的抗惊厥剂或抗癫痫剂 ,通过选择性地阻断电压门控Na+通道,稳定突触前神经元膜并抑制谷氨酸释放。Lamotrigine hydrate 可用于研究癫痫、局灶性癫痫等神经性疾病。
T37847 Zonisamide-13C2,15N

Zonisamide-13C2,15N

Zonisamide-13C2,15N is intended for use as an internal standard for the quantification of zonisamide by GC- or LC-MS. Zonisamide is an antiepileptic agent.1 It selectively inhibits the repeated firing of sodium channels (IC50 = 2 μg/ml) in mouse embryo spinal cord neurons and inhibits spontaneous channel firing when used at concentrations greater than 10 μg/ml.2 In rat cerebral cortex neurons, zonisamide (1-1,000 μM) inhibits T-type calcium channels with a maximum reduction of 60% of the calcium...

化合物

Anticonvulsant agent 2
Cat.No: T73586
Synonym:
Target: Others
Anticonvulsant agent 1
Cat.No: T10027
Synonym: 4-(2,2-Difluoroethenyl)-α-ethyl-2-oxo-1-pyrrolidineacetamide
Target: Others
N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea
Cat.No: T12156
Synonym:
Target: Others
3-Methyl-GABA
Cat.No: T22509
Synonym:
Target: Others
Lamotrigine hydrate
Cat.No: T60492
Synonym:
Target:
Zonisamide-13C2,15N
Cat.No: T37847
Synonym: Zonisamide-13C2,15N
Target:
Cat. No. Product Name Target Signaling Pathways
T20587 2-Acetonaphthone

2-萘乙酮,beta-Acetylnaphthalene,beta-Acetonaphthalene,2Acetylnaphthalene,2-Acetylnaphthalene,2 Acetylnaphthalene,beta-Naphthyl methyl ketone

Endogenous Metabolite Metabolism
2-Acetonaphthone (beta-Naphthyl methyl ketone) 是内源性代谢产物的一种。

天然产物

2-Acetonaphthone
Cat.No: T20587
Synonym: 2-萘乙酮,beta-Acetylnaphthalene,beta-Acetonaphthalene,2Acetylnaphthalene,2-Acetylnaphthalene,2 Acetylnaphthalene,beta-Naphthyl methyl ketone
Target: Endogenous Metabolite
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