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抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T1005 Amoxicillin

Amoxycillin,阿莫西林

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T1005L Amoxicillin trihydrate

Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。
T6385 Amoxicillin Sodium

阿莫西林钠,Clavulanate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin Sodium (Clavulanate) 是一种有广谱抗菌活性,口服吸收好的抗生素。它能抑制细胞壁中多肽的生物合成,可抑制细胞生长。
T23732 Amoxicillin, L-

L-Amoxicillin,Amoxicillin trihydrate impurity B,Amoxicillin related compound B

Amoxicillin, L- is an antibiotic. It is also useful for the treatment of a number of bacterial infections.
T10306 Amoxicillin D4

Amoxycillin D4

Others Others
Amoxicillin D4 (Amoxycillin D4) is a deuterium-labeled Amoxicillin. Amoxicillin is an antibiotic with broad-spectrum antimicrobial activity.
T33225 m-Chloro-amoxicillin

m-Chloro-amoxicillin is a bioactive chemical.
T78628 Amoxicillin-clavulanate potassium

Antibiotic Microbiology/Virology
Amoxicillin-clavulanate potassium为具备广泛抗菌谱的复合抗生素,潜在应用于研究多种细菌感染。
T73956 Amoxicillin trihydrate mixture with potassium clavulanate (4:1)

Amoxicillin (trihydrate) mixture with potassium clavulanate (4:1) 是一种抗生素 (antibiotic),具有优良的口服吸收性及广谱抗菌作用。该化合物通过抑制细胞壁内多肽的生物合成来阻止细胞生长。
T39811 D-4-Hydroxyphenylglycine

4-Hydroxy-D-phenylglycine,D-(-)-4-Hydroxyphenylglycine,D-4-Hydroxyphenylglycine

D-4-Hydroxyphenylglycine (D-(-)-4-Hydroxyphenylglycine) is a crucial raw material in the synthesis of semisynthetic β-lactam antibiotics, including Amoxicillin and Cefadroxil .
T79282 Antibacterial agent 144

Antibacterialagent 144(compound 8e)是一款效能超过氯霉素和阿莫西林的抗菌药物,专门针对具有多重耐药性的金黄色葡萄球菌。该化合物通过破坏细菌的细胞质膜和抑制生物膜形成来发挥作用。Antibacterialagent 144能与HSA紧密结合(Kd=13.2 μM),显示出卓越的杀菌活性。它还能与DNA相结合,形成超分子复合物,有效阻断DNA复制过程。
T83705 BING TFA

Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria

BING是一种来源于日本稻田鱼(O. laptipes)的抗菌肽,由液泡蛋白质分选相关蛋白13D样(Vps13D)衍生而来。对包括耐甲氧西林的金黄色葡萄球菌(MRSA; MICs = 4-64 µg/ml)在内的各种革兰氏阴性和革兰氏阳性细菌都有活性。与氨苄西林、阿莫西林和新霉素共同使用时,对抗铜绿假单胞菌(P. aeruginosa)表现出协同效应,并能抑制大肠杆菌(E. coli)对卡那霉素和氨苄西林的抗药性发展。在体内,BING提高了被鳗弧菌(E. tarda)感染的O. laptipes的生存率。

化合物

Amoxicillin
Cat.No: T1005
Synonym: Amoxycillin,阿莫西林
Target: Antibacterial, Antibiotic
Amoxicillin trihydrate
Cat.No: T1005L
Synonym: Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate
Target: Antibacterial, Antibiotic
Amoxicillin Sodium
Cat.No: T6385
Synonym: 阿莫西林钠,Clavulanate
Target: Antibacterial, Antibiotic
Amoxicillin, L-
Cat.No: T23732
Synonym: L-Amoxicillin,Amoxicillin trihydrate impurity B,Amoxicillin related compound B
Target:
Amoxicillin D4
Cat.No: T10306
Synonym: Amoxycillin D4
Target: Others
m-Chloro-amoxicillin
Cat.No: T33225
Synonym:
Target:
Amoxicillin-clavulanate potassium
Cat.No: T78628
Synonym:
Target: Antibiotic
Amoxicillin trihydrate mixture with potassium clavulanate (4:1)
Cat.No: T73956
Synonym:
Target:
D-4-Hydroxyphenylglycine
Cat.No: T39811
Synonym: 4-Hydroxy-D-phenylglycine,D-(-)-4-Hydroxyphenylglycine,D-4-Hydroxyphenylglycine
Target:
Antibacterial agent 144
Cat.No: T79282
Synonym:
Target:
BING TFA
Cat.No: T83705
Synonym: Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria
Target:
Cat. No. Product Name Target Signaling Pathways
TN4300 Isojacareubin

MAPK; PKC; Antifection Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Microbiology/Virology
Isojacareubin displays potent activity against H. pylori HP40 clinical isolate with MIC 23.9 uM, which is approximately two times greater than that of the standard drug amoxicillin. Isojacareubin is a potent inhibitor of protein kinase C (PKC), suppresses

天然产物

Isojacareubin
Cat.No: TN4300
Synonym:
Target: MAPK, PKC, Antifection
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