Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T63237 |
Acotiamide hydrochloride
|
||
Acotiamide hydrochloride 是选择性的、口服具有活力的、可逆的乙酰胆酶碱酯 (AChE) 抑制剂 (IC50: 1.79 μM),能够提高胃收缩性,加速胃排空延迟,能够用于研究胃动力障碍的功能性消化不良及肠道炎症。 | |||
T2319 |
Acotiamide monohydrochloride trihydrate
Acotiamide hydrochloride,YM-443 HCl,盐酸阿考替胺,Z-338 HCl |
AChE | Neuroscience |
Acotiamide monohydrochloride trihydrate (Z-338 HCl) 是一种首创的、具有口服活性的胃肠动力药。它通过促毒蕈碱受体拮抗作用和乙酰胆碱酯酶(AChE)抑制作用增强肠神经元释放的乙酰胆碱,从而增强胃排空和胃部适应性,有潜力用于功能性消化不良的研究。 | |||
T70122 |
Acotiamide Methyl Ether
|
||
Acotiamide Methyl Ether is a metabolite of Acotiamide -- an acetylcholinesterase inhibitor which has been shown to stimulate gastric motility and improve gastric motility dysfunction in rats. Acotiamide Hydrochloride has also been shown to improve meal-related symptoms of functional dyspepsia. |