Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1941 |
Ac-RYYRWK-NH2
|
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Potent, selective partial agonist peptide for the NOP receptor (Ki = 0.71 nM). Selective over μ, δ and κ opioid receptors (IC50 > 4000 nM). Increases food intake in vivo. | |||
TP1941L1 |
Ac-RYYRWK-NH2 acetate
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Ac-RYYRWK-NH2 acetate 是一种有效的伤害感受素受体 (NOP) 的部分激动剂,它是内源性 ORL1 受体激动剂。 | |||
T40510 |
Ac-RYYRWK-NH2 TFA
Ac-RYYRWK-NH2 TFA |
||
Ac-RYYRWK-NH2 is a highly effective and specific partial agonist for the nociceptin receptor (NOP). It demonstrates a remarkable affinity for rat cortical membranes ORL1, with [3H]Ac-RYYRWK-NH2 exhibiting a Kd value of 0.071 nM. However, it shows negligible affinity towards μ-, κ-, or δ-opioid receptors. |