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Cat. No. Product Name Target Signaling Pathways
T64237 ASB14780

ASB14780 是一种 4-苯氧衍生物,是一种胞质磷脂酶 cPLA2α 抑制剂 (IC50: 20 nM)。
T37842 ASB 14780

Potent and selective cytosolic phospholipase A2 alpha (cPLA2α) inhibitor (IC50 = 20 nM). Selective for cPLA2α over secreted PLA2α (sPLA2α; exhibits no inhibition at 10 μM). Inhibits cPLA2α-dependent inflammatory responses in vitro in guinea pig and human whole-blood assays. Improves diet-induced liver injury and CCl4-induced hepatic fibrosis in vivo. Orally bioavailable.

化合物

ASB14780
Cat.No: T64237
Synonym:
Target:
ASB 14780
Cat.No: T37842
Synonym:
Target:
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