Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T27951 |
LY392098
LY-392098,LY 392098,AMPA receptor modulator-3 |
GluR; iGluR | Membrane transporter/Ion channel; Neuroscience |
LY392098 (AMPA receptor modulator-3) 是 AMPA 受体的变构调节剂,EC50 为 4.4 μM,可用于哺乳动物神经系统的研究。 | |||
T36809 |
UoS 12258
|
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Positive allosteric modulator of AMPA receptors (pEC50 = 5.2 for potentiation of AMPA-mediated currents in vitro). Also potentiates AMPA-mediated synaptic responses in vivo. Improves performance of rats in various learning and memory paradigms Ward et al (2010) Discovery of N-[(2S)-5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide, a novel clinical AMPA receptor positive modulator. J.Med.Chem. 53 5801 PMID:20614889 |Ward et al (2017) Pharmacological characterization of N-[... |