Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1364L |
ALX 40-4C acetate
ALX 40-4C acetate(143413-49-4 free base) |
Apelin receptor; CXCR | Autophagy; GPCR/G Protein; Immunology/Inflammation |
ALX 40-4C acetate 是趋化因子受体 (Ki = 1 μM) 的 CXCR4 抑制剂,可抑制 HIV-1 X4 株的复制。 ALX 40-4C acetate 是 APJ 受体的拮抗剂 (IC50 = 2.9 μM)。 | |||
TP1364 |
ALX 40-4C
|
||
ALX40-4C is a small peptide inhibitor of the chemokine receptor CXCR4 that can inhibit X4 strains of HIV-1. |