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Cat. No. Product Name Target Signaling Pathways
T14151 AKR1C1-IN-1

NADPH Metabolism
AKR1C1-IN-1 是高选择性 AKR1C1抑制剂(Ki:4 nM)。
T19999 1-Tetralol, (S)-

(S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C

Others Others
1-Tetralol, (S)- ((S)-1-Hydroxytetralin) 可在细胞实验中用作 AKR1C1 的底物。
T61485 S07-2010

S07-2010 is a potent pan-AKR1C inhibitor, effectively inhibiting AKR1C3, AKR1C4, AKR1C1, and AKR1C2 with IC50 values of 0.19, 0.36, 0.47, and 0.73 μM, respectively. This compound induces apoptosis in A549/DDP cells and enhances the cytotoxicity of chemotherapeutic agents in drug-resistant cells, making it a viable option for combating drug resistance. Furthermore, S07-2010 significantly inhibits the proliferation of drug-resistant cells [1].

化合物

AKR1C1-IN-1
Cat.No: T14151
Synonym:
Target: NADPH
1-Tetralol, (S)-
Cat.No: T19999
Synonym: (S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C
Target: Others
S07-2010
Cat.No: T61485
Synonym:
Target:
TargetMol Loading
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