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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T14151 AKR1C1-IN-1

NADPH Metabolism
AKR1C1-IN-1 是高选择性 AKR1C1抑制剂(Ki:4 nM)。
T19999 1-Tetralol, (S)-

(S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C

Others Others
1-Tetralol, (S)- ((S)-1-Hydroxytetralin) 可在细胞实验中用作 AKR1C1 的底物。
T22519 5-bromo-3-phenyl Salicylic Acid

Others Others
AKR1C1 inhibitor
T23912 CPSA

CPSA is an effective and selective AKR1C1 inhibitor.
T61485 S07-2010

S07-2010 is a potent pan-AKR1C inhibitor, effectively inhibiting AKR1C3, AKR1C4, AKR1C1, and AKR1C2 with IC50 values of 0.19, 0.36, 0.47, and 0.73 μM, respectively. This compound induces apoptosis in A549/DDP cells and enhances the cytotoxicity of chemotherapeutic agents in drug-resistant cells, making it a viable option for combating drug resistance. Furthermore, S07-2010 significantly inhibits the proliferation of drug-resistant cells [1].

化合物

AKR1C1-IN-1
Cat.No: T14151
Synonym:
Target: NADPH
1-Tetralol, (S)-
Cat.No: T19999
Synonym: (S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C
Target: Others
5-bromo-3-phenyl Salicylic Acid
Cat.No: T22519
Synonym:
Target: Others
CPSA
Cat.No: T23912
Synonym:
Target:
S07-2010
Cat.No: T61485
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2899 Liquiritin

Liquiritigenin-4'-O-glucoside,Liquiritoside,甘草苷

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Liquiritin (Liquiritigenin-4'-O-glucoside) 是一种从甘草中分离出的类黄酮,是一种竞争性的 AKR1C1 抑制剂,对 AKR1C1AKR1C2 和 AKR1C3 的 IC50分别为 0.62 μM,0.61 μM 和 3.72 μM,在体内有效抑制 AKR1C1 介导的孕酮代谢。它是一种抗氧化剂,具有神经保护、抗癌、抗炎的活性。

天然产物

Liquiritin
Cat.No: T2899
Synonym: Liquiritigenin-4'-O-glucoside,Liquiritoside,甘草苷
Target: Reactive Oxygen Species
TargetMol Loading
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