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Cat. No. Product Name Target Signaling Pathways
T4223 Mitapivat

PKR-IN-1

PKM Metabolism
Mitapivat (PKR-IN-1) 是口服具有活性的变构丙酮酸激酶 (pyruvate kinase) 激活剂,其AC50=20 nM。它在广泛的 PKLR 基因型中增加酶活性、蛋白质稳定性和 ATP 水平。它有潜在的恢复 PK 缺乏的糖酵解途径活性的作用。
T69864 CIDD-0067106

CIDD-0067106 is a novel potent and selective antiproliferative agent, inhibiting the activity of the mtorc1 pathway
T69865 Mitapivat sulfate

Mitapivat sulfate, also known as AG-348 sulfate hydrate, is an allosteric activator of Pyruvate Kinase (PK) that may be useful in the treatment of Pyruvate Kinase Deficiency.

化合物

Mitapivat
Cat.No: T4223
Synonym: PKR-IN-1
Target: PKM
CIDD-0067106
Cat.No: T69864
Synonym:
Target:
Mitapivat sulfate
Cat.No: T69865
Synonym:
Target:
TargetMol Loading
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