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Cat. No. Product Name Target Signaling Pathways
T2063 Tyrphostin 23

RG-50810,TX 825,Tyrphostin A23,AG18

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Tyrphostin 23 (AG18) 是一种EGFR 抑制剂,IC50值为35 μM。
T21128 Lansoprazole sulfide

Lansoprazole impurity C,AG-1777,EC 600-451-9,H 225/18,K-1252

Lansoprazole sulfide is an impurity of Lansoprazole, which is a gastric pump inhibitor.
T69196 AG-012986

AG-012986 is a multitargeted cyclin-dependent kinase (CDK) inhibitor active against CDK1, CDK2, CDK4/6, CDK5, and CDK9, with selectivity over a diverse panel of non-CDK kinases. AG-012986 showed antiproliferative activities in vitro with IC(50)s of <100 nmol/L in 14 of 18 tumor cell lines. In vivo, significant antitumor efficacy induced by AG-012986 was seen (tumor growth inhibition, >83.1%) in 10 of 11 human xenograft tumor models. AG-012986 also showed dose-dependent retinoblastoma Ser(795) hy...
T69197 AG-012986 HCl

AG-012986 HCl is a multitargeted cyclin-dependent kinase (CDK) inhibitor active against CDK1, CDK2, CDK4/6, CDK5, and CDK9, with selectivity over a diverse panel of non-CDK kinases. AG-012986 HCl showed antiproliferative activities in vitro with IC(50)s of <100 nmol/L in 14 of 18 tumor cell lines. In vivo, significant antitumor efficacy induced by AG-012986 HCl was seen (tumor growth inhibition, >83.1%) in 10 of 11 human xenograft tumor models. AG-012986 HCl also showed dose-dependent retinoblas...

化合物

Tyrphostin 23
Cat.No: T2063
Synonym: RG-50810,TX 825,Tyrphostin A23,AG18
Target: EGFR
Lansoprazole sulfide
Cat.No: T21128
Synonym: Lansoprazole impurity C,AG-1777,EC 600-451-9,H 225/18,K-1252
Target:
AG-012986
Cat.No: T69196
Synonym:
Target:
AG-012986 HCl
Cat.No: T69197
Synonym:
Target:
TargetMol Loading
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