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Cat. No. Product Name Target Signaling Pathways
T79583 AChE-IN-36

AChE-IN-36,具有0.04 μM的IC50,作为乙酰胆碱酯酶抑制剂,能够调节ROS水平及NRF2基因的表达。
T36639 Donecopride (fumarate hydrate)

Donecopride is a partial agonist of the serotonin (5-HT) receptor subtype 5-HT4E(Ki= 8.5 nM) and an inhibitor of acetylcholinesterase (AChE; IC50= 16 nM).1It is selective for AChE over butyrylcholinesterase (BChE; IC50= 3,530 nM) but does bind to 5-HT2Band sigma-2 (σ2) receptors (Ki= 1.6 nM for both) in a panel of 42 neurotransmitter receptors and transporters. Donecopride induces release of soluble amyloid precursor protein-α (sAPP-α) in COS-7 cells transiently expressing 5-HT4with an EC50value...

化合物

AChE-IN-36
Cat.No: T79583
Synonym:
Target:
Donecopride (fumarate hydrate)
Cat.No: T36639
Synonym:
Target:
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