Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T29522 |
ABT 102
ABT102,CHEMBL398338,ABT-102 |
TRP/TRPV Channel | Membrane transporter/Ion channel |
ABT 102 (CHEMBL398338) 是瞬时受体电位香草素 1 (TRPV1) 受体的选择性拮抗剂。 | |||
T29522L |
(S)-ABT 102
|
TRP/TRPV Channel | Membrane transporter/Ion channel |
N-[(1S)-5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-N'-1H-indazol-4-ylurea 是一种有效的TRPV1拮抗剂,其IC50为123 nM,可阻断capsaicin 对TRPV1的激活。 |