Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78711 |
A011
|
ATM/ATR | DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
A011,作为一种选择性的ataxia-telangiectasia mutated (ATM)抑制剂,其IC50为1.0 nM,能够在与CPT-11联合应用时,诱导Apoptosis及G2/M期细胞周期阻滞,显示出显著的抗肿瘤活性。 |