Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13413 |
Zoniporide hydrochloride hydrate
CP-597396 hydrochloride hydrate |
Others | Others |
Zoniporide hydrochloride hydrate is a potent and selective sodium-hydrogen exchanger type 1 (NHE-1) inhibitor. Zoniporide hydrochloride hydrate inhibits human NHE-1 with IC50 of 14 nM. | |||
T23566 |
Zoniporide dihydrochloride
|
Others | Others |
Sodium-hydrogen exchanger isoform 1 (NHE1) inhibitor | |||
T21996 |
Zoniporide hydrochloride
CP-597396 hydrochloride |
Sodium Channel | Membrane transporter/Ion channel |
Zoniporide hydrochloride 是一种特异性的 NHE-1 抑制剂,IC50 为 14 nM,是其他 NHE 同工型的 >150 倍特异性。 Zoniporide hydrochloride 对人血小板的 NHE-1 依赖性肿胀的 IC50 为 59 nM。 |