Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3107 |
Alvelestat
AZD9668,Avelestat |
Others; Serine Protease | Others; Proteases/Proteasome |
Alvelestat (AZD9668) 是一种口服活性,亲和性和选择性的中性粒细胞弹性蛋白酶 (NE) 抑制剂,pIC50=7.9 nM,Ki=为 9.4 nM,Kd=9.5 nM。 | |||
T3107L | Alvelestat tosylate | ||
Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation. |