Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22534 |
8-Hydroxy-DPAT hydrobromide
7-(二丙基氨基)-5,6,7,8-四氢-1-萘酚氢溴酸盐,8-OH-DPAT hydrobromide |
5-HT Receptor | GPCR/G Protein; Neuroscience |
8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) 是一种选择性5-HT1A 激动剂,pIC50为 8.19。它对 5-HT1结合位点的亚型有近 1000 倍的选择性。 | |||
T4305 |
8-OH-Dpat
8-Hydroxy-DPAT |
5-HT Receptor | GPCR/G Protein; Neuroscience |
8-OH-Dpat (8-Hydroxy-DPAT) 是选择性5-HT 激动剂,对 5-HT1A 的pIC50值为 8.19,对 5-HT7 的Ki 值为 466 nM,对 5-HT1B (pIC50, 5.42) 和 5-HT (pIC50<5) 的作用很弱。 | |||
T28639 | S(-)-8-Hydroxy-DPAT hydrobromide | ||
S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor. | |||
T23218 |
(R)-(+)-8-Hydroxy-DPAT hydrobromide
|
Others | Others |
5-HT1A serotonin receptor agonist |