Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2298 |
ML204
|
TRP/TRPV Channel | Membrane transporter/Ion channel |
ML204 是有效的TRPC4/TRPC5通道选择性抑制剂,相比于 TRPC6 ,对TRPC4/TRPC5通道的选择性高出 19 倍,不影响其他的 TRP 通道和电压门控的钠、钾或 Ca2+通道。 | |||
T24481 |
ML204 hydrochloride
ML204,ML204 HCl,ML-204 |
||
ML204 is a potent inhibitor of the TRPC4 channel. ML204 inhibited TRPC4β-mediated intracellular Ca(2+) rise (IC50: 0.96 μM) and exhibited 19-fold selectivity against muscarinic receptor-coupled TRPC6 channel activation. |