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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T69109 Ellipticine tartrate

Ellipticine tartrate is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
T68788 Ellipticine quinone

Ellipticine quinone, also known as NSC-383230, is a Drp1 inhibitor. rpitor1 and Drpitor1a inhibited the GTPase activity of Drp1 without inhibiting the GTPase of dynamin 1. Ellipticine quinone showed greater potency than the current std. Drp1 GTPase inhibitor, mdivi-​1, (IC50 for mitochondrial fragmentation are (0.06, and 10 μM, resp.)​. Ellipticine quinone suppressed lung cancer tumor growth in a mouse xenograft model. Ellipticine quinone also inhibited mitochondrial ROS prodn., prevented mi...

化合物

Ellipticine tartrate
Cat.No: T69109
Synonym:
Target:
Ellipticine quinone
Cat.No: T68788
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1166 Ellipticine

玫瑰树碱,NSC 71795,Elliptisine

Topoisomerase DNA Damage/DNA Repair
Ellipticine (Elliptisine) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 活性,对白血病、神经母细胞瘤和胶质母细胞瘤有部分活性。
T4614 Ellipticine hydrochloride

Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐

Topoisomerase DNA Damage/DNA Repair
Ellipticine hydrochloride (NSC-71795 (hydrochloride)) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 的活性。

天然产物

Ellipticine
Cat.No: T1166
Synonym: 玫瑰树碱,NSC 71795,Elliptisine
Target: Topoisomerase
Ellipticine hydrochloride
Cat.No: T4614
Synonym: Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐
Target: Topoisomerase
TargetMol Loading
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