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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T71851 5-trans-Prostaglandin E2

5-trans-Prostaglandin E2 accelerates fibrinolysis by enhancing plasminogen activation mediated by tissue-type plasminogen activator. It also inhibits platelet aggregation in human PRP.
T36160 8-iso Prostaglandin E2

8-iso Prostaglandin E2

8-iso PGE2 is one of several isoprostanes produced from arachidonic acid during lipid peroxidation. It is a potent renal vasoconstrictor in the rat. 8-iso PGE2 inhibits U-46619 or I-BOP-induced platelet aggregation with IC50 values of 0.5 and 5 μM, respectively. When infused into the renal artery of the rat at a concentration of 4 μg/kg/min, 8-iso PGE2 decreases the GFR and renal plasma flow by 80% without affecting blood pressure.

化合物

5-trans-Prostaglandin E2
Cat.No: T71851
Synonym:
Target:
8-iso Prostaglandin E2
Cat.No: T36160
Synonym: 8-iso Prostaglandin E2
Target:
Cat. No. Product Name Target Signaling Pathways
T5014 Prostaglandin E2

地诺前列酮,前列腺素 E2,PGE2,Dinoprostone,Prostaglandin E2 (PGE2)

Endogenous Metabolite; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
Prostaglandin E2 (PGE2) 是一种天然激素,参与人体内的各种生理过程,包括平滑肌收缩和放松、调节血管扩张和收缩、调节血压和炎症调节。

天然产物

Prostaglandin E2
Cat.No: T5014
Synonym: 地诺前列酮,前列腺素 E2,PGE2,Dinoprostone,Prostaglandin E2 (PGE2)
Target: Endogenous Metabolite, Prostaglandin Receptor
TargetMol Loading
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