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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T9704 1-Ethynylpyrene

P450 Metabolism
1-Ethynylpyrene 是有效的细胞色素P450 1A1, 1A2和2B1抑制剂,抑制的IC50分别为 0.18,0.32 和 0.04 μM。
T24988 7ETMC

7 ETMC,7-ETMC

7ETMC is a selective Human Cytochrome P450s 1A1 and 1A2 inhibitor. 7ETMC showed IC50s of 0.46 μM and 0.50 μM for P450s 1A1 and 1A2 in the first six minutes, respectively, and did not show any inhibition activity for P450s 2A6 and 2B1 even at the dose of 5

化合物

1-Ethynylpyrene
Cat.No: T9704
Synonym:
Target: P450
7ETMC
Cat.No: T24988
Synonym: 7 ETMC,7-ETMC
Target:
Cat. No. Product Name Target Signaling Pathways
TQ0161 Mulberrin

桑黄酮,Kuwanon C

Others Others
Mulberrin (Kuwanon C) 能够抑制有机阴离子转运多肽 2B1 介导的雌酮-3-硫酸盐摄取(IC50:1.8±1.5 μM)。

天然产物

Mulberrin
Cat.No: TQ0161
Synonym: 桑黄酮,Kuwanon C
Target: Others
TargetMol Loading
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