Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79797 |
PHD-IN-1
|
HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; Metabolism |
PHD-IN-1(compound 80)作为PHD2的抑制剂,显示出 IC50 ≤5 nM 的高效活性。在Caco2-HIFla-HiBiT-clone-1和Hep3B细胞系中进行的EPO Elisa实验中,其EC50值均为2.5 μM。 |