Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T72153 |
Topoisomerase IV inhibitor 1
|
Topoisomerase | DNA Damage/DNA Repair |
TopoisomeraseIV inhibitor 2 (compound 7d) 作为DNA拓扑异构酶IV(TOPO IV)抑制剂,展现出高效的活性,其对TOPO IV的IC50值为0.23 μM,而对DNA促旋酶的IC50为0.43 μM。此外,该化合物在抗菌领域同样表现出较强的能力,对金黄色葡萄球菌Nerman菌株(Staphylococcus aureus Newman)和大肠杆菌ATCC8739的最小抑菌浓度(MIC)分别为0.972 μM和0.608 μM。 |