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Cat. No. Product Name Target Signaling Pathways
T40288 CDK12-IN-4

CDK12-IN-4

CDK12-IN-4, a pyrazolotriazine compound, exhibits potent inhibition of CDK12 by achieving an IC50 value of 0.641 μM, utilizing high ATP levels (2 mM). Notably, CDK12-IN-4 does not impact CDK2/Cyclin E (IC50 > 20 μM) or CDK9/Cyclin T1 (IC50 > 20 μM) under the influence of high ATP (2 mM) levels (WO2021116178A1).

化合物

CDK12-IN-4
Cat.No: T40288
Synonym: CDK12-IN-4
Target:
TargetMol Loading
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