Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7685 |
USP25/28 inhibitor AZ1
AZ1 |
DUB | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination |
USP25/28 inhibitor AZ1 (AZ1) 是一种口服有效,选择性,非竞争性的双重泛素特异性蛋白酶 USP25/28抑制,IC50分别为 0.7 μM 和0.6 μM。它有抗炎和抗肿瘤作用。 | |||
T68668 |
AZ-1
|
||
AZ-1 is an inducer of ABCA1 and apoE. It enhances ABCA1 activity and decreases P2X7 receptor activity. AZ-1 activates endogenous LXR signaling but shows no direct LXRα or LXRβ agonist activity. |