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Cat. No. Product Name Target Signaling Pathways
T10396 ATM Inhibitor-1

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
ATM Inhibitor-1 is a highly potent, selective and orally active ATM inhibito (IC50: 0.7 nM) anti-tumor activity. It shows weak activity against mTOR (IC50, 21 μM), DNAPK (IC50, 2.8 μM), PI3Kα (IC50, 3.8 μM), PI3Kβ (IC50, 10.3 μM), PI3Kγ (IC50, 3 μM) and PI3Kδ (IC50, 0.73 μM).

化合物

ATM Inhibitor-1
Cat.No: T10396
Synonym:
Target: ATM/ATR
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