Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10299 |
AMG PERK 44
|
ERK | MAPK |
AMG PERK 44 is an orally active and selective PERK inhibitor (IC50: 6 nM) and induces autophagy. It has 1000-fold and 160-fold selectivity over GCN2 (IC50: 7300 nM) and B-Raf (IC50 >1000 nM), respectively. |