Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3586 |
Compound 401
2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one |
DNA-PK | DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
Compound 401 (2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one) 是一种可靶向 mTOR 的合成 DNA-PK 抑制剂,IC50为0.28 μM。 |