Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14947 |
CHDI-390576
|
HDAC | Chromatin/Epigenetic; DNA Damage/DNA Repair |
CHDI-390576 is a CNS penetrant class IIa HDAC inhibitor (IC50s: 54 nM, 60 nM, 31 nM, 50 nM for class IIa HDAC4, HDAC5, HDAC7, HDAC9). It shows >500-fold selectivity over class I HDACs (1, 2, 3) and ~150-fold selectivity over HDAC8 and the class IIb HDAC6 isoform. |