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Cat. No. Product Name Target Signaling Pathways
T10407 Gartisertib

ATR inhibitor 2

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
ATR inhibitor 2 is an orally active, ATP-competitive, and selective ATR inhibitor (Ki <150 pM) with antitumor activity. ATR inhibitor 2 potently inhibits ATR-driven phosphorylated checkpoint kinase-1 (Chk1) phosphorylation (IC50: 8 nM).

化合物

Gartisertib
Cat.No: T10407
Synonym: ATR inhibitor 2
Target: ATM/ATR
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