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Cat. No. Product Name Target Signaling Pathways
T12660 (Rac)-BAY1238097

Epigenetic Reader Domain Chromatin/Epigenetic
(Rac)-BAY1238097 is a inhibitor of BET(IC50 of 1.02 μM for BRD4),used in cancer research.
T12660L BAY1238097

Epigenetic Reader Domain Chromatin/Epigenetic
BAY1238097 是一种具有有效性和选择性的溴结构域和末端外基序(BET)抑制剂,具有抗癌活性,在AML (急性髓性白血病) 和MM (多发性骨髓瘤) 模型中表现出较强的抗增殖活性 。BAY1238097 可用于研究晚期难治性恶性肿瘤。
T13442 (R)-BAY1238097

Others Others
(R)-BAY1238097 is the R-isomer with lower activity of BAY1238097. BAY1238097 is a selective BET inhibitor.

化合物

(Rac)-BAY1238097
Cat.No: T12660
Synonym:
Target: Epigenetic Reader Domain
BAY1238097
Cat.No: T12660L
Synonym:
Target: Epigenetic Reader Domain
(R)-BAY1238097
Cat.No: T13442
Synonym:
Target: Others
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