Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78869 | TWIK-1/TREK-1-IN-2 | Potassium Channel | Membrane transporter/Ion channel |
TWIK-1/TREK-1-IN-2(Compound 2g)为特异性TWIK-1/TREK-1抑制剂,其针对TREK-1同二聚体的IC50值为10.13 μM,以及针对TWIK-1/TREK-1异二聚体的IC50为15.5 μM,表现为潜在的抗抑郁化合物。 |