Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16482 |
PF-05085727
|
PDE | Metabolism |
PF-05085727 inhibits PDE2A >4,000-fold selectivity over PDE1 and PDE3-11. PF-05085727 is an effective, selective and brain penetrant inhibitor of cGMP-dependent PDE2A (IC50=2 nM) . |