Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2422 |
PNU-282987
|
AChR | Neuroscience |
PNU 282987 是一种选择性 α7 烟碱型乙酰胆碱受体 (α7 nAChR) 激动剂,Ki 为 26 nM。 | |||
T22401 |
PNU-282987 S enantiomer hydrochloride
(S)-PNU-282987 HCl |
Others | Others |
(S)-PNU-282987 is the absolute stereochemistry form of PNU-282987. PNU 282987, a potent agonist of α7-containing neuronal nicotinic acetylcholine receptors (nAChRs) with Ki of 26 nM for the rat receptor, has negligible activity against α1β1γδ and α3β4 nAC | |||
T60437 |
PNU-282987 free base
|
||
PNU-282987 (free base) (Compound C7) 是 α7 烟碱乙酰胆碱受体 (nAChR) 的有效激动剂 (EC50 = 154 nM), 也是5-HT3受体的功能性拮抗剂 (IC50 = 4541 nM)。PNU-282987 (free base) 可用于研究中枢和周围神经系统[1]。 | |||
T7695 |
PNU-282987 S enantiomer free base
|
AChR | Neuroscience |
PNU-282987 S enantiomer free base 是 PNU-282987 的 S 型对映体,是 α7 烟碱乙酰胆碱受体的激动剂。 |