Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2525 |
Alosetron hydrochloride
Lotronex,盐酸阿洛司琼,GR 68755C,GR 68755,GR 68755X |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Alosetron hydrochloride (GR 68755) 是一种高选择性的 5-HT3 受体拮抗剂,可减轻清醒或麻醉犬直肠扩张的内脏伤害性效应,具有抗炎活性,用于肠易激综合征的研究。它阻断 5HT3 介导的豚鼠肌间和粘膜下神经元的快速去极化,IC50约为 55 nM。 | |||
T21235 |
Alosetron
Lotronex,GR68755,GR-68755,GR 68755,阿洛司琼 |
||
Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only. | |||
T19190 |
Alosetron D3 Hydrochloride
GR-68755C D3 |
Others | Others |
Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor. | |||
T19191 |
Alosetron-d3
Alosetron D3,GR 68755 D3,GR 68755X D3 |
Others | Others |
Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor. |