Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TCA2511 |
11Beta-hydroxyprogesterone
|
Sodium Channel | Membrane transporter/Ion channel |
The progesterone derivatives 11 alpha- and 11 beta-hydroxyprogesterone are potent inhibitors of 11 beta-hydroxysteroid dehydrogenase (isoforms 1 and 2) in vitro and can confer mineralocorticoid activity on corticosterone in the rat in vivo. 11beta-Hydroxyprogesterone acts as a mineralocorticoid agonist in stimulating Na+ absorption in mammalian principal cortical collecting duct cells. |