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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T37475 Cyclic ADP-Ribose (ammonium salt)

cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)

Cyclic ADP-ribose (cADP-ribose) is an endogenous metabolite of NAD+ that mobilizes the release of stored Ca2+ in the endoplasmic reticulum via ryanodine receptors in various cell types.[1],[2],[3],[4],[5] This second messenger is generated via the cADP-ribose synthases CD38 and CD157.[6],[5],[7] cADP-Ribose may also trigger the cell surface Ca2+ influx channel TRPM2 in a temperature-dependent manner.[8] In vitro, cADP-ribose modulates Ca2+ signaling in rat and mouse cardiomyocytes treated with i...

化合物

Cyclic ADP-Ribose (ammonium salt)
Cat.No: T37475
Synonym: cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)
Target:
Cat. No. Product Name Target Signaling Pathways
T19253 Cyclic ADP-​ribose

cADPR

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cyclic ADP-ribose (cADPR) is an effective calcium mobilization second messenger, which is synthesized from NAD + by ADP-ribosyl cyclase. Cyclic ADP-ribose mainly increases cytosolic calcium through Ryanodine receptor-mediated endoplasmic reticulum release

天然产物

Cyclic ADP-​ribose
Cat.No: T19253
Synonym: cADPR
Target: Calcium Channel
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